99% umunyu wa Tianeptine sodium CAS 30123-17-2
Ibisobanuro
INGINGO | STANDARD | IGISUBIZO |
Kugaragara | Ifu yera kugeza umuhondo | Ifu ya kirisiti yera |
Gukemura | Byoroshye gushonga mumazi na methanol na dichloromethane | Guhuza |
Kumenyekanisha | Na IR, Guhuza nibikorwa bisanzwe | Guhuza |
(2) Itanga reaction ya sodium | Guhuza | |
Impanuka A. | ≤0.1% | Ntibimenyekana |
Ibikoresho bifitanye isano | Ikintu cyose cyanduye cyanduye≤0.1% | 0.060% |
Umwanda wose≤0.4% | 0.36% | |
Ibisubizo bisigaye (GC) | Acetidin≤ 0.5% | ND |
Dichloromethane≤ 0.06% | ND | |
Methanol≤ 0.3% | ND | |
Acetone≤ 0.5% | 0.29% | |
Acetonitrile≤0.041% | 0.022% | |
Ethanol≤0.5% | ND | |
N, N-dimethylformamide≤0.088% | ND | |
Amazi | ≤ 5.0% | 3.8% |
Suzuma (HPLC) | 99.0% -101.0% (Kuri anhydrousbasis) | 99,70% |
Gusaba
Sodium ya Tianeptineumunyuni tricyclic antidepressant.Uburyo bwayo bwo kurwanya antidepressant butandukanye nubwa gakondo tricyclic antidepressants.Irashobora kongera reuptake ya 5-HT muri synaptic.Ingaruka zo gutwara HT neuronal.Ntaho bihurira na choline cyangwa reseptor ya adrenergic.Imiti igabanya ubukana isa niy'inyabutatu, ariko kwihanganira ni byiza kuruta ibya tricyclics.Mu kuvura indwara yo kwiheba byoroheje, bitagereranywa cyangwa bikabije, kwiheba kwa neurogeneque na reaction, guhangayika no kwiheba hamwe n’umubiri, cyane cyane kutagira igifu, no guhangayika no kwiheba ku barwayi batewe n'inzoga mu gihe cyo kuva.